Complete GPCR Assay List
G protein-coupled receptors (GPCRs) are proteins possessing seven cell membrane-spanning domains with extracellular ligand binding sites for specific molecules. Interactions with those sites result in modulation of signal transduction pathways involving second messengers such as cAMP, inositol phosphate or calcium which is ultimately translated into a cellular responses. G protein-coupled receptors are involved in many diseases and are targeted therapeutically by half of all modern medicinal drugs.
| Cat# | Assay Type | Assay Class | Assay Name | $/Well (USD) |
|---|---|---|---|---|
| 100-0328 | Binding | Adenosine | A1 (h) | $62.00 |
| 100-0043 | Binding | Adenosine | A2 | $36.00 |
| 100-0003 | Binding | Adenosine | A2A (h) | $62.00 |
| 100-0004 | Binding | Adenosine | A3 | $62.00 |
| 100-0030 | Binding | Adenosine | AD Non selective | $36.00 |
| 100-0100 | Binding | Adrenergic | Alpha 1 Non selective | $36.00 |
| 100-0005 | Binding | Adrenergic | Alpha 1A | $39.00 |
| 100-0006 | Binding | Adrenergic | Alpha 1B | $36.00 |
| 100-0101 | Binding | Adrenergic | Alpha 2 Non selective | $36.00 |
| 100-0007 | Binding | Adrenergic | Alpha 2A (h) | $62.00 |
| 100-0008 | Binding | Adrenergic | Alpha 2B | $44.00 |
| 300-1019 | Cellular | Adrenergic | Alpha 2B, Agonist (h) | $68.00 |
| 300-1020 | Cellular | Adrenergic | Alpha 2B, Antagonist (h) | $68.00 |
| 100-0102 | Binding | Adrenergic | Alpha 2C | $44.00 |
| 100-0009 | Binding | Adrenergic | Alpha 2C (h) | $62.00 |
| 300-0784 | Cellular | Adrenergic | Alpha 2C Agonist (h) | $68.00 |
| 300-0785 | Cellular | Adrenergic | Alpha 2C Antagonist (h) | $68.00 |
| 100-0990 | Binding | Adrenergic | Alpha2b (h) | $62.00 |
| 100-0104 | Binding | Adrenergic | Beta 1 | $44.00 |
| 100-0010 | Binding | Adrenergic | Beta 1 (h) | $62.00 |
| 300-1025 | Cellular | Adrenergic | Beta 1, Agonist (h) | $68.00 |
| 300-1029 | Cellular | Adrenergic | Beta 1, Antagonist (h) | $68.00 |
| 100-0105 | Binding | Adrenergic | Beta 2 | $44.00 |
| 100-0011 | Binding | Adrenergic | Beta 2 (h) | $62.00 |
| 300-0451 | Cellular | Adrenergic | Beta 2 Agonist (h) | $68.00 |
| 300-0452 | Cellular | Adrenergic | Beta 2 Antagonist (h) | $68.00 |
| 100-0325 | Binding | Adrenergic | Beta 3 (h) | $62.00 |
| 100-0103 | Binding | Adrenergic | Beta Non selective | $39.00 |
| 100-0084 | Binding | Angiotensin II | AT1 (h) | $62.00 |
| 100-0107 | Binding | Angiotensin II | AT1 Peripheral | $48.00 |
| 300-1056 | Cellular | Angiotensin II | AT1, Agonist (h) | $68.00 |
| 300-1057 | Cellular | Angiotensin II | AT1, Antagonist | $68.00 |
| 100-0108 | Binding | Angiotensin II | AT2 Central | $48.00 |
| 100-0109 | Binding | Atrial Naturietic Factor | ANP-A | $48.00 |
| 300-0221 | Cellular | Bradykinin | B1 Agonist (h) | $68.00 |
| 300-0283 | Cellular | Bradykinin | B1 Antagonist (h) | $68.00 |
| 100-0012 | Binding | Bradykinin | B2 | $48.00 |
| 300-0222 | Cellular | Bradykinin | B2 Agonist | $68.00 |
| 100-0073 | Binding | Cannabinoid | CB1 (h) | $62.00 |
| 300-1001 | Cellular | Cannabinoid | CB1, Agonist (h) | $68.00 |
| 300-1002 | Cellular | Cannabinoid | CB1, Antagonist (h) | $68.00 |
| 100-0074 | Binding | Cannabinoid | CB2 (h) | $62.00 |
| 300-0800 | Cellular | Chemokine | CCR2 Agonist (h) (Ca2+) | $68.00 |
| 300-0801 | Cellular | Chemokine | CCR2 Antagonist (h) (Ca2+) | $68.00 |
| 300-1003 | Cellular | Chemokine | CXCR2, Agonist (h) | $68.00 |
| 300-1004 | Cellular | Chemokine | CXCR2, Antagonist (h) | $68.00 |
| 100-0114 | Binding | Cholecystokinin | CCK1 (CCKA) | $48.00 |
| 100-0115 | Binding | Cholecystokinin | CCK2 (CCKB) | $48.00 |
| 100-0117 | Binding | Complement | Anaphylatoxin C5aR (h) | $62.00 |
| 300-1021 | Cellular | Complement | C5a, Agonist (h) | $68.00 |
| 100-0118 | Binding | Corticotropin Releasing Factor | CRF Non selective | $48.00 |
| 300-0225 | Cellular | Corticotropin Releasing Factor | CRF1 Agonist (h) | $68.00 |
| 300-0293 | Cellular | Corticotropin Releasing Factor | CRF1 Antagonist (h) | $68.00 |
| 100-0120 | Binding | Dopamine | D1 | $44.00 |
| 100-0016 | Binding | Dopamine | D1 (h) | $62.00 |
| 300-0227 | Cellular | Dopamine | D1 Agonist (h) (cAMP) | $68.00 |
| 300-0755 | Cellular | Dopamine | D1 Agonist (h) (Luciferase) | $68.00 |
| 300-0226 | Cellular | Dopamine | D1 Antagonist (h) (Ca2+) | $68.00 |
| 300-0284 | Cellular | Dopamine | D1 Antagonist (h) (cAMP) | $68.00 |
| 300-0757 | Cellular | Dopamine | D1 Antagonist (h) (Luciferase) | $68.00 |
| 100-0121 | Binding | Dopamine | D2 | $44.00 |
| 300-1047 | Cellular | Dopamine | D2L, Agonist (h) | $68.00 |
| 300-1048 | Cellular | Dopamine | D2L, Antagonist (h) | $68.00 |
| 100-1006 | Binding | Dopamine | D2s (h) | $62.00 |
| 100-0018 | Binding | Dopamine | D3 | $36.00 |
| 100-1005 | Binding | Dopamine | D4.2 (h) | $62.00 |
| 100-0019 | Binding | Dopamine | D4.4 (h) | $62.00 |
| 100-0116 | Binding | Dopamine | DA Non-Selective (Clozapine) | $44.00 |
| 100-0085 | Binding | Endothelin | ETA (h) | $62.00 |
| 100-0124 | Binding | Endothelin | ETB (h) | $62.00 |
| 100-0024 | Binding | GABA-B | GABA-B | $41.00 |
| 100-0130 | Binding | Galanin | Galanin Non selective | $48.00 |
| 100-0786 | Binding | GammaHydroxyButyrate | GHB | $44.00 |
| 100-0756 | Binding | Glutamate (metabotropic) | mGluR1 | $62.00 |
| 100-0405 | Binding | Glutamate (metabotropic) | mGluR5 | $62.00 |
| 100-0034 | Binding | Histamine | H1 | $44.00 |
| 100-0456 | Binding | Histamine | H1 (h) | $62.00 |
| 300-0998 | Cellular | Histamine | H1, Agonist (h) | $68.00 |
| 300-0999 | Cellular | Histamine | H1, Antagonist (h) | $68.00 |
| 100-0086 | Binding | Histamine | H2 | $44.00 |
| 300-1041 | Cellular | Histamine | H2 Agonist (h) (Ca2+) | $68.00 |
| 300-1040 | Cellular | Histamine | H2 Antagonist (h) (Ca2+) | $68.00 |
| 100-0035 | Binding | Histamine | H3 | $44.00 |
| 300-0229 | Cellular | Histamine | Histamine, H2 Agonist (h) (cAMP) | $68.00 |
| 100-0036 | Binding | Leukotriene | LTB4 (BLT) | $48.00 |
| 100-0481 | Binding | Leukotriene | LTB4 (BLT1) (h) | $62.00 |
| 100-0482 | Binding | Leukotriene | LTB4 (BLT2) (h) | $62.00 |
| 300-0296 | Cellular | Leukotriene | LTB4 Agonist (h) | $68.00 |
| 300-0297 | Cellular | Leukotriene | LTB4 Antagonist (h) | $68.00 |
| 300-0298 | Cellular | Leukotriene | LTC4/D4 Agonist (h) | $68.00 |
| 100-0037 | Binding | Leukotriene | LTD4 (CysLT1) | $48.00 |
| 300-0749 | Cellular | Lysophospholipid | LPA2 (EDG4) Agonist (h) | $68.00 |
| 300-0750 | Cellular | Lysophospholipid | LPA2 (EDG4) Antagonist (h) | $68.00 |
| 300-0737 | Cellular | Lysophospholipid | Sphingosine-1-phosphate S1P3 (EDG3) Agonist (h) | $68.00 |
| 300-0738 | Cellular | Lysophospholipid | Sphingosine-1-phosphate S1P3 (EDG3) Antagonist (h) | $68.00 |
| 100-0134 | Binding | Melatonin | Melatonin Non selective | $48.00 |
| 100-0135 | Binding | Muscarinic | M Non selective Central | $48.00 |
| 100-0136 | Binding | Muscarinic | M Non selective Peripheral | $44.00 |
| 100-0137 | Binding | Muscarinic | M1 | $39.00 |
| 100-0038 | Binding | Muscarinic | M1 (h) | $62.00 |
| 300-0231 | Cellular | Muscarinic | M1 Agonist (h) (Ca2+) | $68.00 |
| 300-0454 | Cellular | Muscarinic | M1 Antagonist (h) (Ca2+) | $68.00 |
| 100-0138 | Binding | Muscarinic | M2 | $44.00 |
| 100-0039 | Binding | Muscarinic | M2 (h) | $62.00 |
| 100-0139 | Binding | Muscarinic | M3 | $44.00 |
| 100-0040 | Binding | Muscarinic | M3 (h) | $62.00 |
| 300-0455 | Cellular | Muscarinic | M3 Agonist (h) (Ca2+) | $68.00 |
| 100-0041 | Binding | Muscarinic | M4 (h) | $62.00 |
| 100-0042 | Binding | Muscarinic | M5 (h) | $62.00 |
| 100-0044 | Binding | Neurokinin | NK1 | $48.00 |
| 100-0140 | Binding | Neurokinin | NK2 (NKA) (h) | $62.00 |
| 300-1022 | Cellular | Neurokinin | NK2, Agonist (h) (Ca2+) | $68.00 |
| 300-1000 | Cellular | Neurokinin | NK2, Agonist (h) (LF) | $68.00 |
| 300-1023 | Cellular | Neurokinin | NK2, Antagonist (h) | $68.00 |
| 100-0141 | Binding | Neurokinin | NK3 (NKB) | $48.00 |
| 100-0142 | Binding | Neuropeptide Y | NPY Non selective | $44.00 |
| 100-0143 | Binding | Neuropeptide Y | NPY1 (h) | $62.00 |
| 100-0045 | Binding | Neuropeptide Y | NPY2 (h) | $62.00 |
| 100-0144 | Binding | Neurotensin | NT | $48.00 |
| 100-0145 | Binding | Neurotensin | NT (h) | $62.00 |
| 100-0149 | Binding | Opioid | Delta | $44.00 |
| 100-0049 | Binding | Opioid | Delta (DOP,OP1) (h) | $62.00 |
| 100-0150 | Binding | Opioid | Kappa 1 | $44.00 |
| 100-0151 | Binding | Opioid | Mu | $44.00 |
| 100-0051 | Binding | Opioid | Mu (h) | $62.00 |
| 300-0234 | Cellular | Opioid | Mu Agonist (h) (GTPgS) | $68.00 |
| 300-0294 | Cellular | Opioid | Mu Antagonist (h) (GTPgS) | $68.00 |
| 100-0072 | Binding | Opioid | Nociceptin, ORL1 (h) | $62.00 |
| 100-0888 | Binding | Opioid | Nociceptin, ORL1 brain (h) | $62.00 |
| 100-0889 | Binding | Opioid | Nociceptin, ORL1 brain (macaque) | $44.00 |
| 100-1024 | Binding | Opioid | Nociceptin, ORL1 brain (Rabbit) | $44.00 |
| 100-0887 | Binding | Opioid | Nociceptin, ORL1 brain (rat) | $44.00 |
| 300-1045 | Cellular | Opioid | Nociceptin, ORL1, Agonist (h) | $68.00 |
| 300-1046 | Cellular | Opioid | Nociceptin, ORL1, Antagonist (h) | $68.00 |
| 100-0147 | Binding | Opioid | OP Non-selective | $40.00 |
| 100-0148 | Binding | Opioid | OP Non-selective (+Na+) | $44.00 |
| 100-0152 | Binding | Oxytocin | Oxytocin | $62.00 |
| 100-0153 | Binding | Platelet Activating Factor | PAF | $62.00 |
| 300-0236 | Cellular | Platelet Activating Factor | PAF Agonist (h) | $68.00 |
| 300-0981 | Cellular | Prostanoid | Prostaglandin E2 (PGE2) Antagonist (h) | $68.00 |
| 300-0980 | Cellular | Prostanoid | Prostaglandin E2 (PGE2) Agonist (h) | $68.00 |
| 100-0157 | Binding | Purinergic | P2Y | $39.00 |
| 100-0055 | Binding | Purinergic | P2Y (h) | $62.00 |
| 300-0238 | Cellular | Purinergic | P2Y2 Agonist (h) | $68.00 |
| 300-0286 | Cellular | Purinergic | P2Y2 Antagonist (h) | $68.00 |
| 100-0158 | Binding | Serotonin | 5HT Non selective | $39.00 |
| 100-0159 | Binding | Serotonin | 5HT1 Non selective | $41.00 |
| 100-0160 | Binding | Serotonin | 5HT1A | $43.00 |
| 100-0057 | Binding | Serotonin | 5HT1A (h) | $62.00 |
| 300-1011 | Cellular | Serotonin | 5HT1A, Agonist (h) | $68.00 |
| 300-1012 | Cellular | Serotonin | 5HT1A, Antagonist (h) | $68.00 |
| 100-0161 | Binding | Serotonin | 5HT1B | $39.00 |
| 100-0058 | Binding | Serotonin | 5HT1D | $44.00 |
| 100-0162 | Binding | Serotonin | 5HT1D (h) | $62.00 |
| 100-0059 | Binding | Serotonin | 5HT2A | $44.00 |
| 100-0163 | Binding | Serotonin | 5HT2A (h) | $62.00 |
| 300-1054 | Cellular | Serotonin | 5HT2A, Agonist (h) | $68.00 |
| 300-1055 | Cellular | Serotonin | 5HT2A, Antagonist (h) | $68.00 |
| 100-0848 | Binding | Serotonin | 5HT2B (h) | $60.00 |
| 300-1013 | Cellular | Serotonin | 5HT2B Agonist (h) | $68.00 |
| 300-1014 | Cellular | Serotonin | 5HT2B Antagonist (h) | $68.00 |
| 100-0060 | Binding | Serotonin | 5HT2C | $44.00 |
| 300-1008 | Cellular | Serotonin | 5HT2C Agonist (h) | $68.00 |
| 300-1009 | Cellular | Serotonin | 5HT2C Antagonist (h) | $68.00 |
| 100-0062 | Binding | Serotonin | 5HT4 | $41.00 |
| 100-0063 | Binding | Serotonin | 5HT5A (h) | $62.00 |
| 100-0064 | Binding | Serotonin | 5HT6 (h) | $62.00 |
| 100-0065 | Binding | Serotonin | 5HT7 (h) | $62.00 |
| 100-0165 | Binding | Somatostatin | SOM Non selective | $48.00 |
| 100-0070 | Binding | Thromboxane | TXA2 (h) | $62.00 |
| 100-0169 | Binding | Thyrotropin Releasing Hormone | TRH | $48.00 |
| 100-0170 | Binding | Vasoactive Intestinal Peptide | VIP Non selective | $48.00 |
| 100-0171 | Binding | Vasopressin | V1 | $48.00 |
| 100-0172 | Binding | Vasopressin | V1A (h) | $62.00 |
| 100-1028 | Binding | Vasopressin | V2 (h) | $62.00 |
| 300-1015 | Cellular | Vasopressin | V2, Agonist (h) | $68.00 |
| 300-1016 | Cellular | Vasopressin | V2, Antagonist (h) | $68.00 |